Drug Development Approaches for Poorly Soluble Compounds

Drug Development Approaches for Poorly Soluble Compounds

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10 different strategies for overcoming poor solubility in drug candidates, drawing on case studies from current drug development projects.

1. Drug development approaches for poorly soluble compounds
2. Solid dispersion technique to improve solubility and, thereby, bioavailability
3. Nanosizing of drugs to improve the apparent dissolution and bioavailability
4. Pharmaceutical Co-crystals
5. Self-micro emulsifying and self-emulsifying drug delivery systems to improve solubility and bioavailability
6. Liposomes and mixed micelles for improvement of drug solubility
7. Improvement of solubility and bioavailability of poorly soluble drugs using mesoporous silica particles
8. Gastrointestinal Dissolution and Absorption of BCS Class II Drugs
9. Cyclodextrin-Based Formulations to Improve Solubility of poorly soluble drugs
10. Cosolvent-based formulations to improve solubility and bioavailability
11. First in-animal studies and formulation considerations
12. Improving aqueous solubility of drug candidates through structural modifications
1. Drug development approaches for poorly soluble compounds
2. Solid dispersion technique to improve solubility and, thereby, bioavailability
3. Nanosizing of drugs to improve the apparent dissolution and bioavailability
4. Pharmaceutical Co-crystals
5. Self-micro emulsifying and self-emulsifying drug delivery systems to improve solubility and bioavailability
6. Liposomes and mixed micelles for improvement of drug solubility
7. Improvement of solubility and bioavailability of poorly soluble drugs using mesoporous silica particles
8. Gastrointestinal Dissolution and Absorption of BCS Class II Drugs
9. Cyclodextrin-Based Formulations to Improve Solubility of poorly soluble drugs
10. Cosolvent-based formulations to improve solubility and bioavailability
11. First in-animal studies and formulation considerations
12. Improving aqueous solubility of drug candidates through structural modifications
ISBN 9783527354788
Media type Book
Edition number 1. Auflage
Copyright year 2026
Publisher Wiley-VCH
Language English